CURRICULUM VITAE

NAME: Mohamed Mohamed Baraka

Birth Date: January 09, 1959

NATIONALITY: Egyptian

CURRENT POSITION:

Assistant professor of Medicinal Chemistry

Department of Medicinal Chemistry, Faculty of Pharmacy,

Zagazig University, Zagazig, Egypt.

MOBIL: 01006887334

PHONE: 0552346529(HOME)

FAX : 0552303266(work)

E-MAIL:

MARITAL STATUS married with four children

EDUCATION:

*Ph.D. In Pharmaceutical Science (Pharmaceutical Chemistry), Ukraine (1992).

Title: SYNTHESIS, PHYSICO-CHEMICAL PROPERTIES AND BIOLOGICAL ACTIVITIES OF 6-CHLORO-7-NITROACREDINE DERIVATIVES

*M.Sc. In Pharmaceutical Science (Pharmaceutical Chemistry) Faculty of

Pharmacy Zagazig University, 1986.

Title: NEW METHODS FOR DETERMINATION OF SOME ANTIRHUMATIC COMPOUNDS.

*B.S. In Pharmaceutical Science (Very Good with Degree of Honor) Faculty of

Pharmacy, Zagazig University, May, 1981.

ACADEMIC POSITION:

Assistance professor of Medicinal Chemistry, Faculty of

Pharmacy, Zagazig University, 2001 tell now.

SCIENTIFIC EXPERIENCE AND SCHOLARSHIP:

1-Research fellowship, Institute of Pharmacy, Kharhov, Ukraine, 1988-1992.

2-Teaching assistant, Faculty of Pharmacy, Zagazig University, 1986-1988.

3-Demonstrator in Medicinal Chemistry Department, Faculty of Pharmacy,

Zagazig University, 1982-1986.

TEACHING EXPERIENCE:

1- Visiting professor of Medicinal Chemistry to Gar younis(Bengazi) and Omar – Almokhtar (Derna)Universities (Libya).

2- Teaching standard courses offered to the fourth and fifth year students of pharmacy emphasis on uses, synthesis, correlation of structure and biological activity for compounds of medicinal and pharmaceutical importance.

3- Teaching and course coordinator of quality Control & Drug analysis course for

fifth year students and for clinical pharmacy students

4- Teaching standard courses of Drug Design as elective course offered to the fifth

year students and clinical pharmacy students

5-Teaching laboratory courses for identification, quantitative and qualitative

assay for drugs in their pure forms and in their pharmaceutical dosage forms.

ORAL EXAMINATION FOR STUDENTS:

1- External examiner for Pharmacy students of [Cairo, Alexandria, Asuot, Ein shams, Mansoura, Tanta, Helwan, Sues Canal, Al-Azhar, 6-October. MSA and El- Menia Universities]

2- External examiner for students of Gar younis and Al -Fateh Universities (Libya).

RESEARCH EXPERIENCE:

1- High experience in using different spectrophotometric techniques in determination and stability indicating assay of drugs in their pure and pharmaceutical dosage forms.

2- Good experience in Synthesis, SAR and study of the biological activity of Anthranilic acid derivatives, Acridines and acridine analogs, Quinazolindione, Pyrazol and thizol derivatives

3- Good experience in use and interpretation of instrumental data, including UV,IR and 1HNMR spectroscopy.

SUPERVISION OF M.SC. THESES IN THE FIELD OF MEDICINAL CHEMISTRY.

1-Synthesis of Some New Quinazolindione Derivatives for Pharmacological Study

2- Instrumental Methods for Determination of Some Antihypertensive Drugs

3- Synthesis and biological screening of new quinazolin-4-(3H) –one derivatives

4- Synthesis and biological evaluation of some heterocyclic compounds

5- Different instrumental techniques for analysis of some gastrointestinal tract drugs

TRAINING COURSES /WORKSHOPS:

1-Workshop in High Performance Liquid Chromatography: Principles and Applications held in Medical Research Institute, Alexandria University, Egypt, July 12, 2005.

2-Workshop in Challenges in Higher Education and Scientific Research Forum:

Supreme Council Universities, Cairo,Egypt, March 21, 2006.

3-Workshop in Quality Assurance and Accreditation (QAAP): Supreme Council Universities, Cairo, Egypt, Nov. 20, 2006.

4-Training course on “Teaching with Technology” Zagazig University, Egypt,

August 5-7/ 8/2006.

5-Training course on “Course Design” Zagazig University, Egypt, Jan 1-2, 2006

6- Training course on “Quality Assurance” Zagazig University, Egypt, May,24- 25, 2006.

7 -Training course on “Problem solving and decision making” Zagazig University, Egypt, May,18-21,2005

8- Training course on“Job ethics” Zagazig University, Egypt, July,24-26 ,2005

9- Training course on “ Teaching Evaluation“ Zagazig University, Egypt,July,4- 7,2007

CONFERENCES:

1-Egeyption Pharmaceutical Society XXXI Conference of Pharmaceutical

Science, Cairo, Egypt, Dec.23, 2008.

2- Al-Azhar 4th International Conference of Pharmaceutical and Biological Sciences, Cairo, Egypt, Feb.13, 2006.

3-Egeyption Pharmaceutical Society XXIX Conference of Pharmaceutical

Science, Cairo, Egypt, Dec.24, 2004.

4-Egeyption Pharmaceutical Society XXVIII Conference of Pharmaceutical Science, Cairo, Egypt, Dec.17, 2002.

5-The first Congress of Early Childhood Mellfare in Sharkia Governorate,Zagazig,

University, Egypt, April,18, 2002.

6- Al-Azhar 2nd International Conference of Pharmaceutical and Biological Sciences,

Cairo, Egypt, Dec.19, 2001.

7- The 3rd Annual Meeting of the Association of Colleges of Pharmacy in the Arab World,Cairo, Egypt, Oct. 14, 1999.

ACTIVITIES:

1-Active member in the Developmental and Appraisal Unit, Faculty of Pharmacy, Zagazig University.2005-2009.

2-Supervisor of the Cultural Committee of Students Union, Faculty of Pharmacy 1994-2003 and 2006-2010.

3-Coordinator of the Higher General Relations Committee of Zagazig University 2002-2003.

4-Coordinator of the Higher Cultural Committee of Zagazig University 2001- 2002.

5- Shared in the selection and decisions regarding various equipment for the

Pharmaceutical Chemistry Department's, Pharmaceutical Consultant Unit and

laboratories Central.

6-Head of and a member of various decision committees for purchasing laboratory equipments

7- Active member of the Accreditation Project "CIQAP". of the Quality

Assurance Unit- Faculty of Pharmacy, Zagazig University.

8- Head of organization committee of graduation day in 2008 and 22010.

9- Head of organization committee of the student training program held in faculty of

pharmacy Zagazig university 21-23 Sept.2010.

10- As a member of the research group working on " achieved the Search and synthesis of new antivirus and anti-inflammatory agents in Egypt funded by , Zagazig, University.

PERSONAL SKILLS:

1- Strong organizational and people management skills

2-Ability to work independently as well as in a team, flexible approach to

advance the work of the research team as well as my own project

3- Hard working

MEMBERSHIP HELD

1-Active member of the Zagazig University Staff Members Club, 1992-2011

2-Member of Consultant Committee of Cultural Population in Sharkiah 2005-2007

5-Cultural Coordinator between Zagazig University and Cultural Population in Sharkiah, 2005

3-Member of the Egyptian Pharmaceutical Society since (1992-present).

4 -Member of the Egyptian Syndicate of Pharmacists (1981-present).

5- Member of the Sharkia Syndicate of Pharmacists (1981-present).

6- Member of the Egyptian Society for Biological Sciences and their Application (2004- present).

7- Member of El-Rowaad Club

REFERENCES:

1-Prof .Dr. Mohamed El-Husseiny El-Sadek, Prof. of Medicinal Chemistry,Faculty of Pharmacy ,Zagazig University, Egypt (Mobil.:002010263394)

3- Prof. Dr. Abel Monem Ateya, Prof. of Pharmacognosy and Director of Unit of Quality Assurance and Accreditation Parameters (QAAP) , Faculty of Pharmacy ,Zagazig).University, Egypt. E-mail: (monem ).

PUBLICATIONS:

(1) SPECTROPHOTOMETRIC METHOD FOR THE DETERMINATION OF FLUFENAMICAND MEFENAMIC ACIDS.

Afaf Aboul Khier, Mohamed El-Sadek and Mohamed M. Baraka

Pharm. Chem. Dept., Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.

Analyst, 112, 1399 (1987).

(2) CLORIMETRIC DETERMINATION OF FLUFENAMIC AND MEFENAMIC ACID

VIA THEIR COMPLEXATION WITH IRON (III).

El-Sadek M., Baraka M.M. and About Khier A

Pharm. Chem. Dept., Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.

Indian Journal of Pharm. Sci. 49, 97 (1987).

(3)DETERMINATION OF DICLOFENAC SODIUM THROUGH THE FORMATION
OF CHARGE TRANSFER COMPLEX WITH CHLORANIL.

M. El-Sadek, M.M. Baraka and About Kheir A

Pharm. Chem. Dept., Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.

Egypt. J. Pharm. Sci. 29, 367 (1988).

(4) SYNTHESIS AND BIOLOGICAL ACTIVITY OF COPPER COMPLEXES OF 4- CHLORO 5-NITRO-N-PHENYLANTHRANILIC ACID DERIVATIVES.

E.E. Meketenka, A.N. Gauaokevitch, T.E Arcenfa, G.B. KazakavandM.M.M. Baraka

Kharkov pharmaceutical institute, Kharkov, Ukraine
Kharkov J. Pharm. Sci. 4, 69 (1991).

(5) STUDY OF CORRELATION DEPENDANC, PHYSICO-CHEMICAL PROPERTIES

AND BIOLOGICAL ACTIVITY OF 4-CHLORO-5-NITRO-N-PHENYLANTHRA-
NILIC ACID DERIVATIVES.

A.N. gaudokevitch, E.N. Cvechnekova, E.E. MEKETENKA, T.A. Kostena
and M.M. Baraka

Kharkov pharmaceutical institute, Kharkov, Ukraine

J. Org. Chem. 29,1578 (1993).

(6)MICRODETERMINATION OF SOME ANALGESICS AND ANTIINFLAMMATORY DRUGS USING SILVER NITRATE.

Hawa M. Khail, Magda M. El-Henawee and *Mohamed M. Baraka

Anal. Chem. Dept. and *Med. Chem. Dept, Faculty of Pharmacy, Zagazig
University, Zagazig, Egypt.

Zagazig J. Pharm. Sci. 4, 40 (1995).

(7) SPECTROSCOPIC METHODS FOR THE DETERMINATION OF FLURBIPOFEN
AND TIAPROFENIC ACID.

Mohamed M. Baraka*, Magda M. El-Henawee and Hawa M. Khalil

*Med. Chem. Dept., and Anal. Chem. Dept., Faculty of Pharmacy, Zagazig
University, Zagazig, Egypt.

Zagazig J. Pharm. Sci. 5,138 (1996).

(8) A NOVEL APPROACH TO ISOQUINOLOINE SYNTHESIS.

* Mohamed I. Al-Asmawi, Osamal. El-Sabbagh and Mohamed M. Baraka

* Org. Chem. Dept. and Med. Chem. Dept, Faculty of Pharmacy, Zagazig
University, Zagazig, Egypt.

Bull. Fac. Pharm., Cairo Univ. 38, 13 (2000).

(9)SYNTHESIS OF NOVAL 2,4-(1H.3H)-QUINAZOLINEDIONE DERIVATIVES
WITH ANALGESIC AND ANTI-INFLAMMATORY ACTIVITIES.

Mohamed M. Baraka

Med. Chem. Dept., Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.

Bull.Fac.Pharm.Cairo Univ.,:vol38.No.1.92000).

(10) SPECTROPHOMETRIC DETERMINATION OF CARBOCISTEINE AN FAMOTIDINEIN IN THEIR DOSAGE FORMS.

Mohamed M. Baraka, Sobhy M. El-AdI, Osama I. El-Sabbagh

Med. Chem. Dept., Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.

Bull. Fac. Pharm. Cairo Univ. 38, 163 (2000).

(11) SPECTROPHOMETRIC DETERMINATION OF DOMPERIDONE.

Sobhy M. El-AdI, Mohamed M. Baraka and *Gamal H. Ragab

Med. Chem. Dept., and *Anal. Chem. Dept., Faculty of Pharmacy, Zagazig
University, Zagazig, Egypt.

Alex. J. Pharm. Sci. 14, 134 (2000).

(12) SPECTROPHOMETRIC DETERMINATION OF MELATONIN IN PURE AND IN
IN PHARMACEUTICAL PREPARATIONS.

Mohamed M. Baraka and Sobhy M. El-AdI

Med. Chem. Dept., Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.

Alex. J. Pharm. Sci. 14,123 (2000).

(13) SYNTHESIS AND EVALUATION OF SOME NEW 2,4-(1H,3H)-QUINAZOLINEDIONE DERIVATIVES AS POTENTIAL ANALGESIC AND ANTIINFLAMMATORY AGENTS

Mohamed El-sadek,Mohamed M.M.Baraka, Samia M.Mostafa*and Mostafa Kh.Soltan.

Medicinal Chemistry Department ,Faculty of Pharmacy, Zagazig University Zagazig, Egypt *Pharm. Chem. Dept. Faculty of Pharmacy , Suez Canal University, Ismaelia, Egypt.

Egypt. J. Pharm. Sci., 44, No. 1, pp. 87-99 (2003).

(14) SYNTHES OF SOME 2,4-(1H,3H)-QUINAZOLINE-DIONE WITH ANALGESIC AND ANTI-INFLAMMATORY ACTIVITY

Mohamed El-sadek, ,Samia M.Mostafa,* Mohamed M.Baraka and Mostafa Kh.Soltan.

Medicinal Chemistry Department ,Faculty of Pharmacy, Zagazig University Zagazig, Egypt *Pharm. Chem. Dept. Faculty of Pharmacy , Suez Canal University, Ismaelia, Egypt.

Al-azhar. j . Pharm. Sci . 33,pp.9-19 March (2006)

(15) SPECTROPHOTOMETRIC DETERMINATION OF RAMIPRIL, ENALAPRIL MALEATE AND FOSINOPRIL THROUGH REACTION WITH 2,4-DINITRO

PHENYLHYDRAZINE AND CHARGE-TRANSFERE COMPLEXATION WITH CHLORANIL

Mohamed M. Baraka,*aMohamed El Sadek,*Ewais Moussa M. Moussa** and Nashat M. M. Abd-Alaty**

* Medicinal Chemistry Department, Faculty of Pharmacy, Zagazig University, Zagazi

** Nuclear Materials Authority, Cairo, Egypt.

Bull.Fac.Pharm. Cairo Univ.Vol.46,No.1pp.153-161(2008).

(16) SPECTROPHOTOMETRIC AND ATOMIC ABSORPTION DETERMINATION

OF RAMIPRIL,ENALAPRIL MALEATE AND FOSINOPRIL THROUGH

TERNARY COMPLEX FORMATION WITH MOLYBDENUM (V)- THIOCYANATE

*a Mohamed Mohamed BARAKA, *Mohamed EL-SADEK, ** Ewais Moussa Mohamed MOUSSA and **Nashat Mohamed Alanowar ABD-ALATY

* Medicinal Chemistry Department, Faculty of Pharmacy, Zagazig University, P.C.44519, Zagazig.

** Nuclear Materials Authority, P.O.Box 530 Almady, Cairo, Egypt.

Bull.Chem.Pharm.Vol.56 (11) 1521-1527(2008) Japan

(17)SYNTHESIS AND ANTIVIRAL ACTIVITY OF NEW PYRAZOLE AND THIAZOLE

DERIVATIVES

Osama I. El-Sabbagh a,*, Mohamed M. Baraka a, Samy M. Ibrahim a, Christophe Pannecouque b, Graciela Andrei b, Robert Snoeck b, Jan Balzarini b, Adel A. Rashad a

a Department of Medicinal Chemistry, Faculty of Pharmacy, Zagazig University, Zagazig,

Egypt

b Rega Institute for Medical Research, Faculty of Medicine, K.U. Leuven, Leuven, Belgium

European Journal of Medicinal Chemistry 44 (2009) 3746–3753.

(18) DESGIN, SYNTHESIS AND PRELIMINARY ANTIVIRAL SCREENING OF NEW

N- PHENYLPYRAZOLE AND DIHYDROISOXAZOLE DERIVATIVES

A. A. Rashad, O. I. El-Sabbagh, Mohamed M. Baraka, S. M. Ibrahim, C.

Pannecouque*, G. Andrei*, R. Snoeck *,J. Balzarini*, A. Mostafa**

Department of Medicinal Chemistry, Faculty of Pharmacy, Zagazig University,44511,

Zagazig, Egypt.

*Rega Institute for Medical Research, Faculty of Medicine, K.U. Leuven, Leuven,

Belgium

*Environmental Virology Laboratory, Department of Water Pollution, National Research

Centre, Dokki, Egypt

Med. Chem. Res.(2010)19:1025-1035, DOI 10.1007/s00044

(19) SYNTHESIS OF NEW 2,3-DIHYDROQUINAZOLIN-4(1H)-ONE DERIVATIVES

FOR ANALGESIC AND ANTI-INFLAMMATORY EVALUATION

Osama I. El-Sabbagh, Samy M. Ibrahim, Mohamed M. Baraka, Hend Kothayer

Department of Medicinal Chemistry, Faculty of Pharmacy, Zagazig University, 44511

Zagazig,Egypt.

Archiv der Pharmazie Chem. Life Sci. Vol. 343 (5), 274-281(2010)

(20) COLORIMETRIC DETERMINATION OF EZETIMIBE IN PURE FORM

AND IN PHARMACEUTICAL PREPARATION

Mohamed M.Baraka* , Hawa M. Khalil** and Khairia M. Al-Ahmary***

*Department o Medicinal Chemistry, Faculty of Pharmacy ,zagazig university , zagazig, Egypt.

** Department of Chemistry, Girl collage of Education, King Khalid University, Abha, Kingdom of Saudi Arabia.

*** Department of Chemistry, Girl collage of Education, King Abdull Aziz University, Jeddah, Kingdom of Saudi Arabia.

Bull. Fac. Pharm. Cairo Univ., Vol. 46, No. 1 (2008)

(21)COLORIMETRIC DETERMINATION OF RAMIPRIL, ENALAPRIL MALEATE AND

FOSINOPRI IN THEIR PHARMACEUTICAL FORMULATIONS

*Mohamed El Sadek, *aMohamed M.Baraka **Ewais Moussa M. Moussa and **Nashat M. M. Abd-Alaty

*Medicinal Chemistry Department, Faculty of Pharmacy, Zagazig

University, P.C.44519 Zagazig

**Nuclear Materials Authority, P.C.530 Almaady, Cairo, Egypt.

Egypt.J. pharm.Sci.50, pp.95-109(2009)

(22)Synthesis of new benzotriazepin-5(2H)-one derivatives of expected antipsychotic

Activity

Samy M. Ibrahim, Mohamed M. Baraka, Osama I. El-Sabbagh, Hend

Kothayer

DOI 10.1007/s00044-012-0102-2

Medicinal Chemistry Research 22:1488-1496(2013)

1