Indian Patent Journal

Granted Patents-July-2009

Bulk Drugs & Intermediates

S.No. / Patent Number / Application Number / Date of Application / Date of Priority / Title of Invention / Name of Patentee / Date of Publication of Abstract u/s 11(A) / Date of Publication of Patent Grant
1 / 213,200 / 883/MUMNP/2005 / 13/01/2004 / 13/01/2003 / A PROCESS OF MANUFACTURING ESTERS AND ETHERS OF PROBUCOL OR SALTS THEREOF / ATHEROGEN ICS, INC., USA / 21/10/2005 / 3/7/2009
2 / 235,390 / 1217/KOLNP/2005 / 24/12/2003 / 24/12/2002 / (R)-2-AMINO-1,4-DIHYDRO-6- METHYL-4-(3-NITROPHENYL)-3,5-PYRIDINEDICARBOXYLIC ACID 3-(1- DIPHENYLMETHYLAZETIDIN-3-YL) ESTER 5-ISOPROPYL ESTER OR A PHARMACOLOGICALLY ACCEPTABLE SALT THEREOF / SANKYO COMPANY, LIMITED., UBE INDUSTRIES,LTD., JAPAN / 03/11/2006 / 3/7/2009
3 / 235,392 / 1341/KOLNP/2004 / 24/03/2003 / 01/04/2002 / SUBSTITUTED PIPERAZINE COMPOUNDS . / ELI LILLY AND COMPANY, USA / 14/07/2006 / 3/7/2009
4 / 235,407 / 608/KOLNP/2004 / 05/11/2002 / 08/11/2001 / NOVEL1,2,4-THIADIAZOLIUM DERIVATIVES AS MELANOCORTIN RECEPTOR MODULATORS / ORTHO-MCNEIL PHARMACEUTICAL CORPORATION, USA / 21/04/2006 / 3/7/2009
5 / 234,667 / 498/DEL/2003 / 27/03/2003 / A PROCESS FOR THE PRODUCTION OF ACYLATED PRODUCTS BY REDUCTIVE ACYLATION OF NITRO, AZIDO AND CYANO ARENES / COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH, INDIA / 09/03/2007 / 10/7/2009
6 / 234,832 / 822/DELNP/2004 / 29/12/2003 / 29/12/2003 / PRIMERS FOR IDENTIFICATION OF ARTEMISININ PRODUCING PLANTS / COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH, INDIA / 04/08/2006 / 10/7/2009
7 / 234,856 / 3471/DELNP/2005 / 25/03/2004 / 26/03/2003 / "A METHOD FOR PREPARING A 2- SUBSTITUTED-5- OXO-3- PYRAZOLIDINECA RBOXYLATE COMPOUND OF FORMULA I" / E.I. DU PONT DE NEMOURS AND COMPANY, USA / 17/08/2007 / 10/7/2009
8 / 234,912 / 2911/DELNP/2004 / 03/04/2003 / 09/04/2002 / "COMPOSITION FOR CELL PROLIFERATION" / OTSUKA PHARMACEUTI CAL CO., LTD., JAPAN / 25/05/2007 / 10/7/2009
9 / 234,974 / 3320/DELNP/2005 / 31/03/2003 / 31/03/2003 / "NOVEL NITRILE GLYCOSIDE USEFUL AS A BIO- ENHANCER OF DRUGS AND NUTRIENTS" / COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH, INDIA / 31/08/2007 / 10/7/2009
10 / 234,975 / 4039/DELNP/2005 / 13/03/2004 / 13/03/2003 / "PROTEIN CONJUGATE HAVING PROLONGED IN VIVO HALF-LIFE" / HANMI PHARM. CO., LTD., REPUBLIC OF KOREA / 24/08/2007 / 10/7/2009
11 / 234,977 / 1183/DEL/1997 / 07/05/1997 / "PHENYL - PIPERAZINYL ALKYLAMINO COMPOUNDS HAVING THE FORMULA I, PHARMACEUTICAL COMPOSITION
AND PROCESS FOR PREPARING THE SAME" / JANSSEN PHARMACEUTICA N. V., BELGIUM / 11/03/2005 / 10/7/2009
12 / 235,042 / 917/DEL/1997 / 09/04/1997 / 10/04/1996 / "SUBSTITUTED [2- (1-PIPERAZINYL) ETHOXY] METHYL COMPOUNDS OF FORMULA (I)" / UCB, S.A., BELGIUM / 11/03/2005 / 10/7/2009
13 / 235,045 / 2924/DELNP/2004 / 16/12/2002 / 16/12/2002 / A PROCESS FOR PREPARING BREVIFOLIOL / COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH, INDIA / 13/07/2007 / 10/7/2009
14 / 235,086 / 4659/DELNP/2005 / 26/04/2004 / 28/04/2003 / "A 4,4-DIFLUORO-1,2,3,4- TERAHYDRO-5H- 1-BENZAZEPINE COMPOUND " / ASTELLAS PHARMA INC., JAPAN / 17/08/2007 / 10/7/2009
15 / 233,964 / 260/MUM/2006 / 24/02/2006 / IMPROVED PROCESS FOR THE PREPARATION OF PHENYL FLUORENOL / MR. SAXENA ALOK, INDIA / 13/04/2007 / 10/7/2009
16 / 234,324 / IN/PCT/2001/01628/ MUM / 27/06/2000 / 02/07/1999 / ANTIPSYCHOTIC CYCLIC N-ARALKYL AMINES / SANOFI- SYNTHELABO, FRANCE / 01/04/2005 / 10/7/2009
17 / 234,330 / 495/MUMNP/2006 / 21/10/2003 / 21/10/2003 / NOVEL METHOD FOR PREPARATION OF CRYSTALLINE PERINDOPRIL ERBUMINE / LUPIN LIMITED, INDIA / 24/08/2007 / 10/7/2009
18 / 234,415 / 1208/MUM/2006 / 31/07/2006
16:07:38 / PROCESS FOR MANUFACTURE OF 2- (2-FLUOROBIPHENYL) PROPIONIC ACID (FLURBIPROFEN) / FDC Limited, INDIA / 08/12/2006 / 10/7/2009
19 / 234,427 / 1015/MUMNP/2006 / 01/02/2005 / 05/02/2004 / SUBSTITUTED THIENO-AND THIAZOLO -[2, 3-D] PYRIDINES AS INHIBITORS OF TIE2 / ASTRAZENECA AB, SWEDEN / 29/06/2007 / 10/7/2009
20 / 234,466 / 341/MUMNP/2005 / 29/11/1999 / 27/11/1998 / NONSTEROIDAL ANTIINFLAMMATORI ES / SCHERING AKTIENGESELL SCHAFT, GERMANY / 30/09/2005 / 10/7/2009
21 / 234,470 / 1140/MUM/2004 / 26/10/2004 / PARENTERAL FORMULATION / M/S. LYKA LABORATORIES LIMITED, INDIA / 02/02/2007 / 10/7/2009
22 / 234,764 / 848/MUMNP/2006 / 20/12/2004 / 22/12/2003 / NOVEL COMPOUNDS / ASTRAZENECA AB, SWEDEN / 18/05/2007 / 10/7/2009
23 / 234,841 / 639/MUM/2003 / 18/06/2003 / 26/06/2002 / PREPARATION OF COLOURLESS DIBENZYLAMINE / LANXESS DEUTSCHLAND GMBH, GERMANY / 11/02/2005 / 10/7/2009
24 / 234,843 / 271/MUM/2005 / 11/03/2005 / AN IMPROVED PROCESS OF GLIMEPIRIDE / IPCA LABORATORIES LTD., INDIA / 20/07/2007 / 10/7/2009
25 / 234,844 / 399/MUM/2004 / 31/03/2004 / IMPROVED PROCESS FOR PREPARATION OF RECOMBINANT HUMAN GRANULOCYTE COLONY STIMULATING
FACTOR IN PICHIA PASTORIS / RELIANCE LIFE SCIENCES PRIVATE LIMITED, INDIA / 08/06/2007 / 10/7/2009
26 / 234,848 / 340/MUMNP/2005 / 21/02/2001 / 23/02/2000 / COMPOUND OF GENERAL FORMULA (A) / UCB FARCHIM S A ( AG-LTD), SWITZERLAND / 30/09/2005 / 10/7/2009
27 / 234,872 / IN/PCT/2002/00672/ MUM / 12/01/2001 / 14/01/2000 / 1,2
BIARYLBENZIMIDAZ OLES AND THEIR PHARMACEUTICAL USE / SCHERING AKTIENGESELL SCHAFT, GERMANY / 28/02/2004 / 10/7/2009
28 / 234,873 / 1301/MUMNP/2005 / 23/12/2002 / 28/12/2001 / TETRAHYDROQUINOL INE ANALOGUES AS MUSCARINIC AGONISTS / ACADIA PHARMACEUTI CALS INC, USA / 12/05/2006 / 10/7/2009
29 / 234,922 / 271/MUM/2006 / 27/02/2006 / IMPROVED PROCESS FOR PREPARING ROSUVASTATIN CALCIUM SALT / CADILA HEALATHCARE LIMITED, INDIA / 26/10/2007 / 10/7/2009
30 / 234,924 / 114/MUM/2003 / 30/01/2003 / 13/02/2002 / CONTINUOUS ADIABATIC PROCESS FOR NITRATING / LANXESS DEUTSCHLAND GMBH, GERMANY / 04/02/2005 / 10/7/2009
31 / 234,930 / IN/PCT/2002/00200/ MUM / 28/08/2000 / 26/08/1999 / A PROCESS FOR THE PREPARATION OF SPHERICAL AGGLOMERATES OF TELITHROMYCIN CRYSTALS / AVENTIS PHARMA S A, FRANCE / 13/01/2006 / 10/7/2009
32 / 234,991 / 91/MUM/2005 / 28/01/2005 / AN IMPROVED PROCESS FOR THE PREPARATION OF THYMIDINE DERIVATIVE / EMCURE PHARMACEUTI CALS LTD, INDIA / 21/09/2007 / 10/7/2009
33 / 235,003 / 1265/MUM/2005 / 07/08/2005 / CONTINENT OSTOMY DEVICE / JAGAD RAJAN BHANDRAKUMAR, INDIA / 28/10/2005 / 10/7/2009
34 / 235,011 / 495/MUMNP/2005 / 24/05/2000 / 10/12/1997 / PROCESS FOR PREPARING A NOVEL ECHINOCANDIN COMPOUND OF FORMULA II / AVENTIS PHARMA S.A, FRANCE / 07/10/2005 / 10/7/2009
35 / 235,553 / 1513/KOLNP/2004 / 30/04/2003 / 01/05/2002 / PROCESS FOR PREPARING 6- ALKYLIDENE PENEM DERIVATIVES . / WYETH, USA / 08/12/2006 / 10/7/2009
36 / 235,586 / 473/KOLNP/2005 / 12/09/2003 / 16/09/2002 / PYRAZOLO[3,4- B]PYRIDINE COMPOUNDS, AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS. / GLAXO GROUP LIMITED, UK / 09/06/2006 / 10/7/2009
37 / 234,339 / 3595/CHENP/2005 / 29/06/2004 / 30/06/2003 / PROCESS FOR PREPARING 3- ACYLAMNOBENZ OFURAN-2- CARBOXYLIC ACID DERIVATIVE / MITSUBISHI TANABE PHARMA CORPORATION, Japan / 25/05/2007 / 17/7/2009
38 / 234,342 / 1237/CHENP/2004 / 07/06/2004 / 06/12/2001 / IMIDAZOQUINOLI NES COMPOUNDS / 3M INNOVATIVE PROPERTIES COMPANY, USA / 10/02/2006 / 17/7/2009
39 / 234,346 / 274/CHENP/2006 / 22/07/2004 / 22/07/2003 / 3, 4- DISUBSTITUTED 1H-PYRAZOLE COMPOUNDS AND THEIR USE AS CYCLIN DEPENDENT KINASES (CDK) AND GLYCOGEN SYNTHASE KINASE-3 (GSK-3) MODULATORS / ASTEX THERAPEUTICS LIMITED, UK / 06/07/2007 / 17/7/2009
40 / 234,347 / 1146/CHENP/2006 / 01/10/2004 / 03/10/2003 / BICYCLO'3.1.1HEPT ANE SUBSTITUTED BENZIMIDAZOLON E AND QUINAZOLINONE DERIVATIVES AS AGONISTS ON HUMAN OR L1 RECEPTORS / SOLVAY PHARMACEUTIC ALS B.V, Netherlands / 31/08/2007 / 17/7/2009
41 / 234,360 / 922/CHE/2004 / 14/09/2004 / AN IMPROVED PROCESS FOR THE PREPARATION OF AN
INTERMEDIATE FOR ANTI- ALZHEMIER DRUG DONEPEZIL HYDROCHLORIDE / NATCO PHARMA LIMITED, INDIA / 02/03/2007 / 17/7/2009
42 / 234,363 / 1042/CHENP/2006 / 25/08/2004 / 27/08/2003 / A PROCESS FOR PRODUCING AN AROMATIC UNSATURATED COMPOUND / SUMITOMO CHEMICAL COMPANY LIMITED, Japan / 29/06/2007 / 17/7/2009
43 / 234,365 / 239/CHENP/2004 / 02/07/2002 / 06/07/2001 / A PROCESS FOR THE PREPARATION OF STATIN DERIVATIVES / CIBA HOLDING INC., Germany / 12/09/2005 / 17/7/2009
44 / 234,366 / 270/CHE/2004 / 24/03/2004 / NOVEL CONDENSED PYRIMIDONES / ORCHID RESEARCH LABORATORIES LTD, INDIA / 02/12/2005 / 17/7/2009
45 / 234,367 / 376/CHENP/2004 / 23/08/2002 / 24/08/2001 / A PROCESS FOR PREPARING A GLYCOPEPTIDE PHOSPHONATE DERIVATIVE OF FORMULA I / THERAVANCE, INC., USA / 23/12/2005 / 17/7/2009
46 / 234,371 / 1965/CHENP/2004 / 31/10/2002 / 07/02/2002 / PRODUCTION METHOD OF (R)-3- HYDROXY-3-(2- PHENYLETHYL) HEXANOIC ACID AND INTERMEDIATE THEREOF / SUMITOMO CHEMICAL COMPANY LIMITED, Japan / 24/02/2006 / 17/7/2009
47 / 234,372 / 2122/CHENP/2006 / 14/12/2004 / 15/12/2003 / A PROCESS FOR PREPARING 2,3- CIS-SUBSTITUTED 2- ARYLPROPENALS / BASF AKTIENGESELL SCHAFT, Germany / 06/07/2007 / 17/7/2009
48 / 234,376 / 3617/CHENP/2005 / 04/05/1999 / 11/05/1998 / BENZALDOXIM COMPOUNDS / BASF AKTIENGESELL SCHAFT, Germany / 14/09/2007 / 17/7/2009
49 / 234,377 / 2373/CHENP/2005 / 26/03/2004 / 27/03/2003 / A COMPOSITION COMPRISING OF TRIGLYCERIDES USEFUL IN NORMALIZATION OF INFRADIAN RHYTHM / SUNTORY LIMITED, USA
R.T. VANDERBILT COMPANY, INC / 31/08/2007 / 17/7/2009
50 / 234,400 / 2854/CHENP/2006 / 19/01/2005 / 04/02/2004 / SUBSTITUTED DIUREA COMPOUNDS / ACTIVE BIOTECH AB, Sweden / 06/07/2007 / 17/7/2009
51 / 234,401 / 794/CHENP/2006 / 23/07/2004 / 08/09/2003 / THIENOPYRAZOLE S / AVENTIS PHARMACEUTI CALS INC., USA / 08/06/2007 / 17/7/2009
52 / 234,402 / 2271/CHENP/2005 / 05/03/2004 / 18/03/2003 / 2-(BUTYL-1- SULFONYLAMINO)
-N-[1(R)-(6- METHOXYPYRIDIN
-3-YL)-PROPYL]- BENZAMIDE, AND PHARMACEUTICA L PREPARATIONS
CONTAINING SAID
COMPOUND / SANOFI- AVENTIS DEUTSCHLAND GMBH, GERMANY / 20/07/2007 / 17/7/2009
53 / 234,405 / 934/CHENP/2006 / 17/09/2004 / 19/09/2003 / PROCESS FOR ENANTIOSELECTI VE SYNTHESIS OF SINGLE ENANTIOMERS OF MODAFINIL BY ASYMMETRIC OXIDATION / CEPHALON FRANCE / 15/06/2007 / 17/7/2009
54 / 234,408 / 515/CHENP/2006 / 10/08/2004 / 11/08/2003 / CEPHALOSPORIN ACYLASE MUTANT AND METHOD FOR PREPARING 7-ACA USING SAME / SANDOZ AG, SWITZERLAND / 06/07/2007 / 17/7/2009
55 / 234,409 / 155/CHENP/2006 / 15/07/2004 / 15/07/2003 / A PROCESS FOR THE MANUFACTURE OF TETRAZOLE DERIVATIVE / NOVARTIS AG, SWITZERLAND / 29/06/2007 / 17/7/2009
56 / 234,523 / 299/CHENP/2006 / 23/07/2004 / 25/07/2003 / NOVEL DIBENZO[B,F]OXE PINE-10- CARBOXAMIDES AND PHARMACEUTICA L USES THEREOF / NOVARTIS AG, SWITZERLAND / 06/07/2007 / 17/7/2009
57 / 234,567 / 1425/CHENP/2006 / 27/10/2004 / 28/10/2003 / A PROCESS FOR PREPARING ANTIHYPERGLICE MIC THIAZOLIDINEDIO NE COMPOUND PIOGLITAZONE, ROSIGLITAZONE AND TROGLITAZONE / SANDOZ AG, SWITZERLAND / 06/07/2007 / 17/7/2009
58 / 234,625 / 105/CHE/2004 / 11/02/2004 / NOVEL PROCESS FOR THE PREPARATION OF BETA- POLYMORPHIC FORM OF IMATINIB MESYLATE / NATCO PHARMA LTD, INDIA / 02/03/2007 / 17/7/2009
59 / 234,634 / 2748/CHENP/2006 / 24/12/2004 / 26/12/2003 / 1,2- DI(CYCLIC)SUBSTI TUTED BENZENE COMPOUNDS / EISAI CO., LTD. JAPAN / 08/06/2007 / 17/7/2009
60 / 234,639 / 1019/CHENP/2006 / 24/09/2004 / 26/09/2003 / PYRIDYLACETYLENES AND COMPOSITIONS THEREOF / NOVARTIS AG, SWITZERLAND / 29/06/2007 / 17/7/2009
61 / 234,660 / 3185/CHENP/2005 / 29/04/2004 / 29/04/2003 / N-EPSILON AND N- ALPHA DERIVATIZED HISTIDINE AND METHOD FOR PREPARING THE SAME / UNIVERSITY OF ZURICH, Switzerland / 01/06/2007 / 17/7/2009
62 / 234,661 / 2247/CHENP/2005 / 12/03/2004 / 14/03/2003 / SUBSTITUTED ANILINE DERIVATIVES / H. LUNDBECK A/S, DENMARK / 31/08/2007 / 17/7/2009
63 / 234,742 / 490/CHENP/2006 / 25/06/2004 / 09/07/2003 / SUBSTITUTED TETRACYCLINE COMPOUNDS / PARATEK PHARMACEUTI CALS, INC., USA / 18/05/2007 / 17/7/2009
64 / 234,746 / 356/CHENP/2006 / 29/07/2004 / 29/07/2003 / PYRIDYL DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS / XENON PHARMACEUTI CALS INC, Canada / 06/07/2007 / 17/7/2009
65 / 234,750 / 3087/CHENP/2005 / 14/05/2004 / 21/05/2003 / BENZOTHIAZOL CARBAMIC ACID ESTERS OF THE GENERAL FORMULA I / F. HOFFMANN LA ROCHE AG, SWITZERLAND / 20/07/2007 / 17/7/2009
66 / 234,751 / 805/CHENP/2006 / 18/06/2004 / 18/06/2004 / NOVEL ANALOGS OF 3-O-ACETYL-11- KETO-B- BOSWELLIC ACID / GOKARAJU, Ganga, Raju, GOKARAJU, Rama, Raju,GOTTUMU KKALA, Venkata, Subbaraju,GOLA KOTI, Trimurtulu, INDIA / 08/06/2007 / 17/7/2009
67 / 234,754 / 2347/CHENP/2005 / 18/03/2004 / 21/03/2003 / SUBSTITUTED P- DIAMINOBENZENE DERIVATIVES / H. LUNDBECK A/S, DENMARK / 31/08/2007 / 17/7/2009
68 / 234,757 / 3411/CHENP/2005 / 09/06/2004 / 17/06/2003 / CIS-IMIDAZOLINES AS MDM2 INHIBITORS / F. HOFFMANN LA ROCHE AG, SWITZERLAND / 08/06/2007 / 17/7/2009
69 / 234,766 / 885/CHE/2004 / 02/09/2004 / A PROCESS FOR THE PREPARATION OF ESCITALOPRAM FROM 5- IODOPHTHALIDE / NATCO PHARMA LIMITED, INDIA / 29/09/2006 / 17/7/2009
70 / 234,767 / 3058/CHENP/2005 / 05/05/2004 / 19/05/2003 / BENZIMIDAZOLE-
2-CARBOXYLIC AMIDES AS FACTOR Xa INHIBITORS / SANOFI- AVENTIS DEUTSCHLAND GMBH, Germany / 08/06/2007 / 17/7/2009
71 / 234,785 / 163/CHENP/2004 / 11/06/2002 / 29/06/2001 / AMINE COMPOUNDS AND CURABLE COMPOSITIONS DERIVED THEREFROM / VIRGINIA TECH INTELLECTUAL PROPERTIES, INC, USA / 09/12/2005 / 17/7/2009
72 / 234,866 / 3189/CHENP/2006 / 18/02/2005 / 02/03/2004 / PROCESS FOR THE PREPARATION OF TRYPTASE INHIBITORS / AVENTIS PHARMACEUTI CALS INC., USA / 08/06/2007 / 17/7/2009
73 / 234,890 / 240/CHENP/2007 / 20/07/2005 / 21/07/2004 / AN IN-VITRO METHOD OF DISTINGUISHING TUBERCULOSIS MODELS / CENTRE FOR DNA FINGERPRINTIN G AND DIAGNOSTICS [CDFD], INDIA / 24/08/2007 / 17/7/2009
74 / 234,898 / 758/CHE/2003 / 22/09/2003 / PROCESS FOR THE PREPARATION OF STERILE CEPHALOSPORIN / ORCHID CHEMICALS & PHARMACEUTI CALS LTD, INDIA / 18/11/2005 / 17/7/2009
75 / 235,115 / 1470/CHENP/2005 / 02/12/2003 / 04/12/2002 / NOVEL FUSED 1,3- DIHYDRO- IMIDAZOLE RING COMPOUNDS HAVING DPPIV- INHIBITING ACTIVITIES / EISAI R & D MANAG EMENT COMPANY LTD. JAPAN / 22/06/2007 / 17/7/2009
76 / 235,127 / 2311/CHENP/2005 / 10/02/2004 / 19/02/2003 / METHOD OF RECRYSTALLISIN G A CYCLIC BENZAMIDINE DERIVATIVE / EISAI R & D MANAGEMENT CO. LTD, JAPAN / 28/11/2008 / 17/7/2009
77 / 235,207 / 1087/CHENP/2006 / 16/08/2004 / 30/09/2003 / PRODUCTION PROCESS OF OPTICALLY PURE
2- (4- HYDROXYPHENOX Y) - PROPIONIC ACID COMPOUNDS / SYNGENTA LIMITED, UK / 17/08/2007 / 17/7/2009
78 / 235,208 / 349/CHENP/2006 / 27/07/2004 / 29/07/2003 / PROCESS FOR PRODUCING IMIDE COMPOUND / DAINIPPON SUMITOMO PHARMA CO., LTD., JAPAN / 06/07/2007 / 17/7/2009
79 / 235,212 / 1567/CHENP/2006 / 05/11/2004 / 07/11/2003 / PROCESS FOR THE PREPARATION OF A TRIFLUOROMETH YLTHIOETHER / CHEMINOVA A/S, Denmark / 06/07/2007 / 17/7/2009
80 / 235,214 / 1565/CHENP/2006 / 05/11/2004 / 06/11/2003 / AMIDOACETONITR ILE DERIVATIVES / NOVARTIS AG, SWITZERLAND / 06/07/2007 / 17/7/2009
81 / 235,240 / 3409/CHENP/2005 / 08/06/2004 / 17/06/2003 / CIS-2,4,5-TRIARYL-IMIDAZOLINES / F. HOFFMANN-LA ROCHE AG, SWITZERLAND / 12/12/2008 / 17/7/2009
82 / 235,247 / IN/PCT/2002/1142/ CHE / 18/01/2001 / 28/01/2000 / PROCESS FOR THE PREPARATION OF ACETYL- AMIDINIOPHENYL ALANYL- CYCLOHEXYLGLY CYL- PYRIDINIOALANIN AMIDES / SANOFI AVENTIS DEUTSCHLAND GMBH, GERMANY / 09/03/2007 / 17/7/2009
83 / 235,248 / 2728/CHENP/2005 / 11/03/2004 / 24/03/2003 / BENZENESULFON AMIDE DERIVATIVE OF FORMULA I / ACTIMIS PHARMACEUTI CALS, INC., USA / 08/06/2007 / 17/7/2009
84 / 235,251 / 648/MAS/2002 / 02/09/2002 / AN IMPROVED PROCESS FOR PREPARATION OF CRYSTALLINE FORM-I OF PANTOPRAZOLE SODIUM SESQUIHYDRATE / DR. REDDY'S LABORATORIES LIMITED, INDIA / 03/08/2007 / 17/7/2009
85 / 235,302 / 1892/MAS/1998 / 21/08/1998 / 22/08/1997 / N- AROYLPHENYLAL ANINE DERIVATIVES / F HOFFMANN- LA ROCHE AG, SWITZERLAND / 04/03/2005 / 17/7/2009
86 / 235,323 / 1947/CHENP/2005 / 17/02/2004 / 18/02/2003 / NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS / F. HOFFMANN- LA ROCHE AG, SWITZERLAND / 28/11/2008 / 17/7/2009
87 / 235,678 / 1636/KOLNP/2005 / 28/01/2004 / 29/01/2003 / THIENOPYRIMIDINE COMPOUNDS AND USE THEREOF . / TAKEDA PHARMACEUTICAL COMPANY LIMITED, JAPAN / 24/11/2006 / 31/7/2009

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Formulations

S.No. / Patent Number / Application Number / Date of Application / Date of Priority / Title of Invention / Name of Patentee / Date of Publication of Abstract u/s 11(A) / Date of Publication of Patent Grant
1 / 235,410 / 1635/KOLNP/2005 / 15/01/2004 / 16/01/2003 / A COMPOSITION COMPRISING SELECTIVE SEROTOTONIN 2A/2C RECEPTOR INVERSE AGNOIST / ACADIA PHARMACEUTI CALS INC, USA / 21/07/2006 / 3/7/2009
2 / 234,521 / 3850/DELNP/2005 / 12/03/2004 / 13/03/2003 / "A COMPOSITION COMPRISING
1,1,1,33,3- PENTAFLUOROBUT ANE (HFC-365mfc) AND 1,1,1,3,3- PENTAFLUOROPRO PANE (HFC-245fa)" / SOLVAY (Societe, Belgium
Anonyme) / 17/08/2007 / 10/7/2009
3 / 234,577 / 192/DELNP/2006 / 17/07/2004 / 29/07/2003 / "PHARMACEUTICA L COMPOSITIONS" / BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG., GERMANY / 10/08/2007 / 10/7/2009
4 / 234,885 / 519/DEL/2003 / 28/03/2003 / "A SYNERGISTIC COMPOSITION USEFUL FOR THE PREPARATION OF IMPROVED SILICON CARBIDE POWDER" / COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH, INDIA / 13/04/2007 / 10/7/2009
5 / 234,977 / 1183/DEL/1997 / 07/05/1997 / "PHENYL - PIPERAZINYL ALKYLAMINO COMPOUNDS HAVING THE FORMULA I, PHARMACEUTICAL COMPOSITION AND PROCESS FOR PREPARING THE SAME" / JANSSEN PHARMACEUTICA N. V., BELGIUM / 11/03/2005 / 10/7/2009
6 / 235,025 / 1172/DEL/2003 / 19/09/2003 / "A PROCESS FOR THE DESIGNING OF PRIMERS USEFUL FOR THE DETECTOPN OF MYCOBACTERIUM TUBERCULOSIS" / INDIAN COUNCIL OF MEDICAL RESEARCH, INDIA / 27/05/2005 / 10/7/2009
7 / 235,026 / 62/DELNP/2006 / 14/07/2004 / 17/07/2003 / "CONTROLLED RELEASE SOFT CAPSULES" / BANNER PHARMACAPS , INC., USA / 24/08/2007 / 10/7/2009
8 / 234,061 / 1221/MUM/2004 / 10/11/2004 / STAVUDINE CONTROLLED RELEASE TABLET / EMCURE PHARAMACEUT ICALS LIMITED, INDIA / 09/06/2006 / 10/7/2009
9 / 234,153 / 517/MUM/2004 / 05/05/2004 / STABLE LIPOSOMAL NEBULIZING INHALATION FORMULATIONS FOR CONTROLLED PULMONARY DELIVERY SYSTEMS / BAJAJ AMRITA,KHALE ANUBHA, INDIA / 29/09/2006 / 10/7/2009
10 / 234,178 / 226/MUMNP/2006 / 30/09/2003 / 30/09/2003 / EXTENDED RELEASE FORMULATION OF ß-LACTAM ANTIBIOTICS / LUPIN LIMITED, INDIA / 29/06/2007 / 10/7/2009
11 / 234,324 / IN/PCT/2001/01628/ MUM / 27/06/2000 / 02/07/1999 / ANTIPSYCHOTIC CYCLIC N-ARALKYL AMINES / SANOFI- SYNTHELABO, FRANCE / 01/04/2005 / 10/7/2009
12 / 234,325 / 1393/MUMNP/2005 / 19/05/2004 / 22/05/2003 / COMPOSITION COMPRISING A PDE4
INHIBITOR AND A PDE5 INHIBITOR / NYCOMED GMBH
ALTANA PHARMA AG, Germany / 06/07/2007 / 10/7/2009
13 / 234,330 / 495/MUMNP/2006 / 21/10/2003 / 21/10/2003 / NOVEL METHOD FOR PREPARATION OF CRYSTALLINE PERINDOPRIL ERBUMINE / LUPIN LIMITED, INDIA / 24/08/2007 / 10/7/2009
14 / 234,422 / 1141/MUMNP/2006 / 18/02/2005 / 09/03/2004 / EYE DROPS CONSISTING OF FILTERED CLAYEY WATER FOR TREATING GLAUCOMA / NEUMANN,Armand, France / 25/05/2007 / 10/7/2009
15 / 234,425 / 1353/MUMNP/2005 / 23/06/2004 / 26/06/2003 / A COMPOSITION FOR INHIBITING THE GROWTH OF ANTIBIOTIC RESISTANT OF BACTERIA BY USING PENTANE-1,5-DIOL / AMBRIA DERMATOLOG Y AB, SWEDEN / 19/05/2006 / 10/7/2009
16 / 234,459 / 563/MUMNP/2005 / 20/07/2001 / 07/04/1999 / 1-PHENACY-3- PHENYL-3- PIPERIDYETHYL COMPOUND FOR USE IN PATHOLOGICAL PHENOMENA INVOLVING TACHYKININ SYSTEM AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME / SANOFI- SYNTHELABO, FRANCE / 07/10/2005 / 10/7/2009
17 / 234,460 / 446/MUM/2005 / 07/04/2005 / PHARMACEUTICAL COMPOSITION CONSISTING OF COX- II INHIBITOR AND MUSCLE RELAXANT / LYKA LABS LIMITED, INDIA / 16/03/2007 / 10/7/2009
18 / 234,461 / 926/MUM/2003 / 08/09/2003 / NOVEL DUAL RELEASE COMBINATION OF A CARDIOVASCULAR DRUG COMPRISING ANTIHYPERTENSIVE AND DIURETIC AGENTS / M/S. IPCA LABORATORIES LIMITED, INDIA / 08/06/2007 / 10/7/2009
19 / 234,470 / 1140/MUM/2004 / 26/10/2004 / PARENTERAL FORMULATION / M/S. LYKA LABORATORIES LIMITED, INDIA / 02/02/2007 / 10/7/2009
20 / 234,478 / 158/MUMNP/2004 / 04/10/2002 / 04/10/2001 / DUAL ACTION ANTIBIOTICES / MORPHOCHEM AKTIENGESELLSCHAFT FÜR KOMBINATORISCHE CHEMIE, GERMANY / 18/02/2005 / 10/7/2009
21 / 234,704 / 819/MUM/2003 / 18/08/2003 / HARD CAPSULE SHELL CONSISTING OF GELATIN AND HYDROXYPROPYL METHYLCELLULOSE AND NOVEL METHOD OF PREPARATION THEREOF / L M COLLEGE OF PHARMACY, INDIA / 18/02/2005 / 10/7/2009
22 / 234,792 / 1425/MUM/2004 / 29/12/2004 / BILAYER TABLETS OF OXCARBAZEPINE FOR CONTROLLED DELIVERY AND A PROCESS OF PREPARATION THEREOF / M/s.J.B.CHEMIC ALS & PHARMACEUTI CALS LTD, INDIA / 21/07/2006 / 10/7/2009
23 / 234,801 / 1301/MUM/2003 / 22/12/2003 / GASTRORETENTIVE SYSTEMS AND NOVEL PHARMACEUTICAL COMPOSITIONS THEREOF / MANGAL SHAILESH NAGARSENKER, INDIA / 20/04/2007 / 10/7/2009
24 / 234,843 / 271/MUM/2005 / 11/03/2005 / AN IMPROVED PROCESS OF GLIMEPIRIDE / IPCA LABORATORIES LTD., INDIA / 20/07/2007 / 10/7/2009
25 / 234,867 / 219/MUMNP/2006 / 01/08/2004 / 31/07/2003 / MICROCAPSULES LOADED WITH
ACTIVE INGREDIENTS AND A METHOD FOR THEIR PREPARATION / SOL-GEL TECHNOLOGIE S LTD, Israel / 29/06/2007 / 10/7/2009
26 / 234,868 / 780/MUM/2003 / 08/08/2003 / NOVEL PARENTERAL FORMULATION FOR PROTON PUMP INHIBITOR / CADILA HEALTHCARE LIMITED, INDIA / 01/04/2005 / 10/7/2009
27 / 234,874 / 1025/MUMNP/2003 / 29/05/2002 / 31/05/2001 / PHARMACEUTICAL COMBINATIONS / ASTRAZENECA AB, SWEDEN / 21/10/2005 / 10/7/2009
28 / 234,910 / IN/PCT/2001/00453/ MUM / 10/05/1999 / 05/06/1998 / A PHARMACEUTICAL COMPOSITION CONTAINING ACE INHIBITORS AND USING MAGNESIUM OXIDE AS STABILIZER / WARNER- LAMBERT COMPANY, USA / 04/03/2005 / 10/7/2009
29 / 234,931 / 1622/MUM/2005 / 26/12/2005 / NOVEL TOPICAL COMPOSITIONS OF SODIUM FUSIDATE / SALGAOCAR DILIP RAMCRISNA, INDIA / 22/09/2006 / 10/7/2009
30 / 234,943 / 510/MUMNP/2003 / 05/12/2001 / 07/12/2000 / PHARMACEUTICAL PREPARATION IN THE FORM OF A SUSPENSION COMPRISING AN ACID LABILE ACTIVE INGREDIENT / ALTANA PHARMA AG, GERMANY / 11/02/2005 / 10/7/2009
31 / 234,967 / 324/BOM/1999 / 29/04/1999 / SUSTAINED RELEASE PHARMACEUTICAL COMPOSITION FOR CONTROLLING ASTHMA / CIPLA LIMITED, INDIA / 18/03/2005 / 10/7/2009
32 / 234,968 / 195/BOM/1999 / 17/03/1999 / THE COMPOSITION FOR TABLETS FOR REDUCING CHOLESTEROL / CIPLA LIMITED, INDIA / 18/03/2005 / 10/7/2009
33 / 234,969 / 181/BOM/1999 / 16/03/1999 / A PHARMACEUTICAL COMPOSITION FOR TOPICAL APPLICATION / CIPLA LIMITED, INDIA / 18/03/2005 / 10/7/2009
34 / 235,060 / 1070/MUM/2002 / 02/12/2002 / AN IMPROVED PHARMACEUTICAL COMPOSITION FOR ASTHMA AND RELATED DISORDERS / CIPLA LIMITED, INDIA / 28/01/2005 / 10/7/2009
35 / 235,145 / 527/MUM/2004 / 07/05/2004 / NOVEL ORAL COMPOSITIONS / SAPTE VINAY RAMAKANT, INDIA / 05/05/2006 / 10/7/2009
36 / 235,522 / 1142/KOLNP/2003 / 11/03/2002 / 30/03/2001 / A MEDICAL AEROSOL FORMULATION FOR INHALATION BASED ON A CARBOXYLIC ACID SALT AS SOLID EXCIPIENT / JAGOTEC AG, SWITZERLAND / 14/10/2005 / 10/7/2009
37 / 235,527 / 741/KOLNP/2005 / 26/09/2003 / 27/09/2002 / A PHARMACEUTICAL GEL PREPARATION / ZENTARIS GMBH, GERMANY / 26/01/2007 / 10/7/2009
38 / 235,531 / 724/KOLNP/2004 / 01/11/2001 / 01/11/2001 / AN EMULSION FOR TOPICAL APPLICATION TO THE SURFACE OF AN EYE AND A PHARMACEUTICAL COMPOSITION / YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM, ISRAEL / 05/12/2008 / 10/7/2009
39 / 235,539 / 688/KOLNP/2006 / 18/10/2004 / 23/10/2003 / CONTROLLED RELEASE STERILE INJECTABLE ARIPIPRAZOLE FORMULATION AND METHOD . / OTSUKA PHARMACEUTICAL CO., LTD., JAPAN / 03/08/2007 / 10/7/2009
40 / 235,540 / 1610/CAL/1998 / 08/09/1998 / 18/09/1997 / WATER SOLUBLE ORGANIC SOLVENT FROM PRODUCTS AND PHARMACEUTICAL FORMULATION . / TEVA PHARMACEUTIC AL WORKS PLC, ISRAEL / 30/09/2005 / 10/7/2009
41 / 235,545 / IN/PCT/2002/1119/ KOL / 16/03/2001 / 20/03/2000 / A PHARMACEUTICAL COMPOSITION, A PHARMACEUTICAL DOSAGE UNIT AND A PHARMACEUTICAL PACK THEREOF . / WYETH, USA / 11/03/2005 / 10/7/2009
42 / 235,552 / 550/KOL/2004 / 08/09/2004 / 10/09/2003 / A COMPOSITION FOR TREATING ACNE, WRINKLES AND FOR REDUCING RETINOID INDUCED REDNESS . / JOHNSON & JOHNSON CONSUMER COMPANIES, INC, USA
., / 06/10/2006 / 10/7/2009
43 / 235,556 / IN/PCT/2001/1209/ KOL / 17/05/2000 / 24/05/1999 / EMULSION VEHICLE FOR POORLY SOLUBLE DRUGS . / SONUS PHARMACEUTIC ALS , INC ., USA / 11/03/2005 / 10/7/2009
44 / 235,579 / 1316/KOLNP/2005 / 16/12/2003 / 19/12/2002 / MEDICINAL COMPOSITION FOR THE PROPHYLAXIS AND TREATMENT OF HYPERGLYCAEMIA. / SIGMA-TAU INDUSTRIE FARMACEUTICH E RIUNITE S.p.A., ITLAY / 09/06/2006 / 10/7/2009
45 / 234,343 / 2264/CHENP/2006 / 20/12/2004 / 23/12/2003 / A PHOSPHATE ESTER OF FLORFENICOL HAVING SUPERIOR WATER SOLUBILITY / SCHERING- PLOUGH LTD., Switzerland / 08/06/2007 / 17/7/2009
46 / 234,362 / 100/CHENP/2006 / 12/07/2004 / 10/07/2003 / A COMPOSITION OF PACKAGED VIRUS LIKE PARTICLES / CYTOS BIOTECHNOLO GY AG, SWITZERLAND / 29/06/2007 / 17/7/2009
47 / 234,406 / 715/CHENP/2006 / 23/06/2004 / 26/08/2003 / A PHARMACEUTICA L LIPOSOMAL FORMULATION FOR PHOTODYNAMIC THERAPY / CERAMOPTEC INDUSTRIES, INC., USA / 22/06/2007 / 17/7/2009
48 / 234,522 / 1049/CHENP/2006 / 30/08/2004 / 29/08/2003 / AN ORAL DOSAGE FORM AND METHOD FOR THE PREPARATION OF THE SAME / LIFECYCLE PHARMA A/S, Denmark / 29/06/2007 / 17/7/2009
49 / 234,623 / 2204/CHENP/2006 / 17/12/2004 / 19/12/2003 / A PHARMACEUTICA L FORMULATION COMPRISING A2A RECEPTOR ANTAGONISTS
ION-PAIRED WITH SODIUM DUCOSATE / SCHERING CORPORATION, USA / 08/06/2007 / 17/7/2009
50 / 234,630 / 3261/CHENP/2005 / 03/06/2004 / 04/06/2003 / ARYL- HETEROAROMATI C PRODUCTS, COMPOSITIONS COMPRISING THEM / AVENTIS PHARMA S A, FRANCE / 14/09/2007 / 17/7/2009
51 / 234,631 / 1179/MAS/1997 / 03/06/1997 / 04/06/1996 / A CONCENTRATED LIQUID FORMULATION HAVING ANTIMICROBIAL ACTIVITY / CIBA SPECIALTY CHEMICALS HOLDING INC., GERMANY / 04/03/2005 / 17/7/2009
52 / 234,701 / 301/MAS/2001 / 09/04/2001 / NEW MONOCYCLIC DERIVATIVES OF ARYL ACIDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICA L COMPOSITIONS CONTAINING THEM / DR. REDDY'S LABORATORIES LTD, INDIA / 01/06/2007 / 17/7/2009
53 / 234,747 / 3368/CHENP/2005 / 10/06/2004 / 13/06/2003 / A PROCESS FOR FORMING CAPSULES / DSM IP Assets B.V, NETHERLANDS / 14/09/2007 / 17/7/2009
54 / 234,753 / 1398/MAS/1997 / 25/06/1997 / 03/07/1996 / GRANULATE FOR THE PREPARATION OF FAST- DISINTEGRATING AND FAST- DISSOLVING COMPOSITIONS / ASTELLAS PHARMA EUROPE B V, NETHERLANDS / 04/03/2005 / 17/7/2009
55 / 234,765 / 957/CHE/2004 / 21/09/2004 / DELAYED RELEASE FORMULATION CONTAINING VENLAFAXINE AND A PROCESS FOR PREPARING THE SAME / NATCO PHARMA LIMITED, INDIA / 29/09/2006 / 17/7/2009
56 / 234,784 / 175/CHENP/2006 / 08/07/2004 / 18/07/2003 / PHARMACEUTICA LY COMPOSITION COMPRISING AZETIDINE DERIVATIVES / AVENTIS PHARMA S A, FRANCE / 18/05/2007 / 17/7/2009
57 / 234,785 / 163/CHENP/2004 / 11/06/2002 / 29/06/2001 / AMINE COMPOUNDS AND CURABLE COMPOSITIONS DERIVED THEREFROM / VIRGINIA TECH INTELLECTUAL PROPERTIES, INC, USA / 09/12/2005 / 17/7/2009
58 / 235,104 / 1635/MAS/1995 / 12/12/1995 / A DENTAL COMPOSITION FOR RELIEVING
DENTIN HYPERSENSITIVIT Y / SUN MEDICAL CO., LTD.,,NOBUO NAKABAYASHI, Japan / 15/06/2007 / 17/7/2009
59 / 235,114 / 1217/CHENP/2004 / 05/11/2002 / 05/11/2001 / A PHARMACEUTICA L FORMULATION OF ANGIOTENSIN- (1-7) / UNIVERSIDADE FEDERAL DE MINAS GERAIS- UFMG, BRAZIL / 10/02/2006 / 17/7/2009
60 / 235,115 / 1470/CHENP/2005 / 02/12/2003 / 04/12/2002 / NOVEL FUSED 1,3- DIHYDRO- IMIDAZOLE RING COMPOUNDS HAVING DPPIV- INHIBITING ACTIVITIES / EISAI R & D MANAG EMENT COMPANY LTD. JAPAN / 22/06/2007 / 17/7/2009
61 / 235,210 / 2901/CHENP/2006 / 14/02/2005 / 12/02/2004 / NEW COMBINATIONS OF AN ANTI EMETIC AGENT AND AN ENKEPHALINASE INHIBITOR / BIOPROJET, France / 08/06/2007 / 17/7/2009
62 / 235,211 / 104/MAS/1998 / 16/01/1998 / 17/01/1997 / 3- HETEROCYCLYL- SUBSTITUTED BENZOYL DERIVATIVES / BASF AKTIENGESELL SCHAFT, Germany / 04/03/2005 / 17/7/2009
63 / 235,216 / 858/MAS/1999 / 30/08/1999 / 01/09/1998 / A PROCESS OF PRODUCING A PHARMACEUTICA L COMPOSITION / F. HOFFMANN LA ROCHE AG, SWITZERLAND / 02/03/2007 / 17/7/2009
64 / 235,243 / IN/PCT/2002/49/CH E / 13/07/2000 / 14/07/1999 / A COMPOSITION FOR TREATMENT OF EXTERNAL SECRETION DISORDERS / SUCAMPO AG, USA / 04/03/2005 / 17/7/2009
65 / 235,337 / 461/CHENP/2003 / 05/10/2001 / 06/10/2000 / A METHOD FOR PRODUCING AN ANTIBODY COMPOSITION / KYOWA HAKKO KOGYO CO. LTD, Japan / 15/04/2005 / 17/7/2009
66 / 235,662 / 92/KOLNP/2004 / 26/07/2002 / 26/07/2001 / A FORMULATION COMPRISING A STRAIN OF LACTOBACILLUS SALIVARIUS / ALIMENTARY HEALTH LIMITED, IRELAND / 03/03/2006 / 31/7/2009
67 / 235,677 / 1467/KOLNP/2004 / 04/04/2003 / 04/04/2002 / A PHARMACEUTICAL COMPOSITION / COLEY PHARMACEUTICAL GMBH, GERMANY / 24/11/2006 / 31/7/2009

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Biotechnology

S.No. / Patent Number / Application Number / Date of Application / Date of Priority / Title of Invention / Name of Patentee / Date of Publication of Abstract u/s 11(A) / Date of Publication of Patent Grant
1 / 234,881 / 524/DEL/2003 / 28/03/2003 / A METHOD FOR PREPARING A MULTIPURPOSE READY-TO-EAT HIGH PROTEIN SOY GRANULES / COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH, INDIA / 13/04/2007 / 10/7/2009
2 / 234,912 / 2911/DELNP/2004 / 03/04/2003 / 09/04/2002 / "COMPOSITION FOR CELL PROLIFERATION" / OTSUKA PHARMACEU TICAL CO.,LTD., JAPAN / 25/05/2007 / 10/7/2009
3 / 234,975 / 4039/DELNP/2005 / 13/03/2004 / 13/03/2003 / "PROTEIN CONJUGATE HAVING PROLONGED IN VIVO HALF-LIFE" / HANMI PHARM. CO., LTD., REPUBLIC OF KOREA / 24/08/2007 / 10/7/2009
4 / 235,025 / 1172/DEL/2003 / 19/09/2003 / "A PROCESS FOR THE DESIGNING OF PRIMERS USEFUL FOR THE DETECTOPN OF MYCOBACTERIUM TUBERCULOSIS" / INDIAN COUNCIL OF MEDICAL RESEARCH, INDIA / 27/05/2005 / 10/7/2009
5 / 235,036 / 1586/DEL/2004 / 20/09/2002 / 20/09/2001 / "COMPOUNDS WHICH INHIBIT THE RELEASE OF INFLAMMATORY CYTOKINES" / THE PROCTER & GAMBLE COMPANY, USA / 16/03/2007 / 10/7/2009
6 / 234,154 / 1211/MUM/2004 / 09/11/2004 / A NOVEL PROCESS FOR PURIFICATION OF HUMAN GROWTH HORMONE / USV LTD., INDIA / 09/06/2006 / 10/7/2009
7 / 234,854 / 397/MUM/2004 / 31/03/2004 / METHOD FOR PRODUCING GRANULOCYTE COLONY STIMULATING FACTOR BY CONSTITUTIVE EXPRESSION / RELIANCE LIFE SCIENCES PRIVATE LIMITED, INDIA / 08/06/2007 / 10/7/2009
8 / 234,873 / 1301/MUMNP/2005 / 23/12/2002 / 28/12/2001 / TETRAHYDROQUINOL INE ANALOGUES AS MUSCARINIC AGONISTS / ACADIA PHARMACEUTI CALS INC, USA / 12/05/2006 / 10/7/2009
9 / 234,913 / IN/PCT/2002/00718/ MUM / 03/06/2002 / 23/12/1999 / AN IMMUNOGENIC PROTEIN IN STERILE FORM. / MEDICAL RESEARCH COUNCIL , INTERNATONAL AIDS VACCINE INITIVE, UNIVERSITY OF NAIROBI, KENYA / 13/03/2004 / 10/7/2009
10 / 235,517 / 1/KOLNP/2004 / 14/06/2002 / 04/07/2001 / DNA SEQUENCE HAVING ANTI- REPRESSOR ACTIVITY / CHROMAGENICS B.V., NETHERLANDS / 31/03/2006 / 10/7/2009
11 / 235,537 / IN/PCT/2001/730/ KOL / 23/12/1999 / 23/12/1998 / A HUMAN MONOCLONAL ANTIBODY THAT BINDS CYTOTOXIC T LYMPHOCYTE ANTIGEN 4(CTLA-4), OR AN ANTIGEN BINDING FRAGMENT THEREOF. / PFIZER INC.,ABGENIX INC., USA / 01/09/2006 / 10/7/2009
12 / 235,581 / 277/KOLNP/2005 / 12/08/2003 / 12/08/2002 / NOVEL IMMUNOGENIC LIPOPEPTIDES COMPRISING T- HELPER AND CYTOTOXIC T LYMPHOCYTE (CTL) EPITOPES. / THE COUNCIL OF THE QUEENSLAND INSTITUTE OF MEDICAL RESEARCH, AUSTRALIA / 06/01/2006 / 10/7/2009
13 / 235,596 / 167/KOLNP/2005 / 19/08/2003 / 19/08/2002 / IMMUNOSTIMULATO RY NUCLEIC ACIDS / COLEY PHARMACEUTIC AL GROUP, INC.,COLEY PHARMACEUTIC AL GMBH, GERMANY / 21/04/2006 / 10/7/2009
14 / 234,340 / 2152/CHENP/2004 / 03/03/2003 / 01/03/2002 / CONJUGATES OF THERAPEUTIC OR CYTOTOXIC AGENTS AND BIOLOGICALLY ACTIVE PEPTIDES / THE ADMINISTRATO RS OF THE TULANE EDUCATIONAL FUND, USA / 03/03/2006 / 17/7/2009
15 / 234,341 / 179/CHENP/2006 / 15/07/2004 / 18/07/2003 / A METHOD OF SCREENING A PAK1 INHIBITOR / SANOFI- AVENTIS DEUTSCHLAND GMBH, GERMANY / 08/06/2007 / 17/7/2009
16 / 234,347 / 1146/CHENP/2006 / 01/10/2004 / 03/10/2003 / BICYCLO'3.1.1HEPT ANE SUBSTITUTED BENZIMIDAZOLON E AND QUINAZOLINONE DERIVATIVES AS AGONISTS ON HUMAN ORL1
RECEPTORS / SOLVAY PHARMACEUTI CALS B.V., Netherlands / 31/08/2007 / 17/7/2009
17 / 234,361 / 3333/CHENP/2005 / 10/06/2004 / 11/06/2003 / ANTIMICROBIAL POLYPEPTIDES / NOVOZYMES A/S, Denmark / 18/05/2007 / 17/7/2009
18 / 234,368 / 375/CHENP/2004 / 23/08/2002 / 24/08/2001 / A PROCESS OF PURIFYING A GLYCOPEPTIDE PHOSPHONATE DERIVATIVE OF FORMULA I / THERAVANCE, INC, USA / 23/12/2005 / 17/7/2009
19 / 234,369 / 374/CHENP/2004 / 23/08/2002 / 24/08/2001 / A PROCESS FOR PREPARING A GLYCOPEPTIDE DERIVATIVE OF FORMULA I / THERAVANCE, INC, USA / 23/12/2005 / 17/7/2009
20 / 234,383 / 202/CHE/2004 / 08/03/2004 / A PROCESS FOR THE SYNTHESIS OF
PHARMACOLOGIC ALLY ACTIVE
(Z/E)- GUGGULSTERONE S / LAILA IMPEX, INDIA / 13/01/2006 / 17/7/2009
21 / 234,384 / 3041/CHENP/2005 / 16/04/2004 / 17/04/2003 / USE OF B7-H3 AS AN IMMUNOREGULAT ORY AGENT / WYETH, USA / 25/05/2007 / 17/7/2009
22 / 234,399 / 785/CHENP/2006 / 03/09/2004 / 05/09/2003 / AN EXPRESSION VECTOR FOR TREATMENT OR PREVENTION OF MELANOMA / SANOFI PASTEUR LIMTED, THERION BIOLOGICS, INC., Canada / 08/06/2007 / 17/7/2009
23 / 234,408 / 515/CHENP/2006 / 10/08/2004 / 11/08/2003 / CEPHALOSPORIN ACYLASE MUTANT AND METHOD FOR
PREPARING 7-ACA USING SAME / SANDOZ AG, SWITZERLAND / 06/07/2007 / 17/7/2009
24 / 234,619 / IN/PCT/2001/515/C HE / 14/09/1999 / 14/09/1998 / RECOMBINANT NEWCASTLE DISEASE VIRUS RNA EXPRESSION SYSTEMS AND VACCINES / MOUNT SINAI SCHOOL OF MEDICINE OF NEW YORK UNIVERSITY, USA / 07/09/2007 / 17/7/2009
25 / 234,658 / 764/CHE/2004 / 04/08/2004 / 06/08/2003 / A NUCLEIC ACID BASED ENCRYPTION AND DECRYPTION METHOD / BIOWELL TECHNOLOGY INC, CHINA
RIXFLEX HOLDING LIMITED / 23/06/2006 / 17/7/2009
26 / 234,659 / 1908/CHENP/2004 / 28/01/2003 / 28/01/2002 / HUMAN MONOCLONAL ANTIBODIES TO PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) / MEDAREX, INC., USA / 30/03/2007 / 17/7/2009
27 / 234,660 / 3185/CHENP/2005 / 29/04/2004 / 29/04/2003 / N-EPSILON AND N- ALPHA DERIVATIZED HISTIDINE AND METHOD FOR PREPARING THE SAME / UNIVERSITY OF ZURICH, ISRAEL / 01/06/2007 / 17/7/2009
28 / 234,756 / 457/CHE/2004 / 14/05/2004 / MYCOBACTERIUM TUBERCULOSIS SPECIFIC PROTEIN AND GENE, AND ITS APPLICATIONS / INDIAN INSTITUTE OF SCIENCE, INDIA / 21/04/2006 / 17/7/2009
29 / 234,774 / IN/PCT/2001/773/C HE / 07/12/1999 / 06/04/2000 / GLP-1
ANALOGUES / SOCIETE DE CONSEILS DE RECHERCHES ETD'APPLICATION S SCIENTIFIQUES SAS ,THE ADMINISTRATO RS OF THE TULANE EDUCATIONAL FUND, France / 27/04/2007 / 17/7/2009
30 / 234,776 / 3049/CHENP/2005 / 19/05/2004 / 19/05/2003 / IMMUNOSUPPRESS ANT COMPOUNDS AND A PHARMACEUTICA
L COMPOSITION COMPRISING THE SAME / IRM LLC, USA / 14/09/2007 / 17/7/2009
31 / 234,866 / 3189/CHENP/2006 / 18/02/2005 / 02/03/2004 / PROCESS FOR THE PREPARATION OF TRYPTASE INHIBITORS / AVENTIS PHARMACEUTI CALS, INC., USA / 08/06/2007 / 17/7/2009
32 / 234,869 / 1185/CHENP/2006 / 06/10/2004 / 08/10/2003 / MODIFIED CEA /B7
VECTORS / SANOFI PASTEUR INC.,THERION BIOLOGICS, INC, CANADA / 17/08/2007 / 17/7/2009
33 / 234,890 / 240/CHENP/2007 / 20/07/2005 / 21/07/2004 / AN IN-VITRO METHOD OF DISTINGUISHING TUBERCULOSIS MODELS / CENTRE FOR DNA FINGERPRINTIN G AND DIAGNOSTICS [CDFD], INDIA / 24/08/2007 / 17/7/2009
34 / 235,113 / 1092/MAS/1995 / 24/08/1995 / 06/09/1994 / SOMATOSTATIN PEPTIDES / NOVARTIS AG, SWITZERLAND / 12/09/2008 / 17/7/2009
35 / 235,114 / 1217/CHENP/2004 / 05/11/2002 / 05/11/2001 / A PHARMACEUTICA L FORMULATION OF ANGIOTENSIN- (1-7) / UNIVERSIDADE FEDERAL DE MINAS GERAIS- UFMG, BRAZIL / 10/02/2006 / 17/7/2009
36 / 235,121 / 2199/MAS/1998 / 01/10/1998 / 02/10/1997 / AN ISOLATED POLYPEPTIDE OF CHLAMYDIA AND ITS GENE SEQUENCE / EMERGENT PRODUCT DEVELOPMENT GAITHERSBURG INC., USA / 04/03/2005 / 17/7/2009
37 / 235,200 / IN/PCT/2002/154/C HE / 05/07/2000 / 07/07/1999 / A METHOD FOR PEPTIDE SYNTHESIS, A COMPOSITION OF PEPTIDE FRAGMENTS AND PEPTIDES MADE THEREBY / TRIMERIS, INC., USA / 27/04/2007 / 17/7/2009
38 / 235,241 / 235/CHENP/2006 / 27/05/2004 / 26/07/2003 / "A METHOD OF IMPROVING EFFICACY OF BIOLOGICAL RESPONSE - MODIFYING PROTEINS AND THE EXEMPLARY MUTEINS" / MEDEXGEN CO.,LTD, Republic of Korea / 17/08/2007 / 17/7/2009
39 / 235,245 / IN/PCT/2001/371/C HE / 11/10/1999 / 16/10/1998 / A PROCESS FOR PREPARING A HIGH PURITY TIBOLONE WITH IMPROVED STABILITY / N.V. ORGANON, Netherlands / 04/03/2005 / 17/7/2009
40 / 235,323 / 1947/CHENP/2005 / 17/02/2004 / 18/02/2003 / NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS / F. HOFFMANN- LA ROCHE AG, SWITZERLAND / 28/11/2008 / 17/7/2009
41 / 235,324 / IN/PCT/2002/134/C HE / 23/06/2000 / 25/06/1999 / "AN ISOLATED NUCLEIC ACID COMPRISING SEQ ID NO.1 AND AN ISOLATED POLYPEPTIDE COMPRISING SEQ ID NO.2" / BASF AKTIENGESELL SCHAFT, Germany / 12/10/2007 / 17/7/2009
42 / 235,336 / IN/PCT/2002/324/C HE / 08/09/2000 / 09/09/1999 / CATIONIC LIPOSOME DELIVERY OF TAXANES TO ANGIOGENIC BLOOD VESSELS / THE REGENTS OF THE UNIVERSITY OF CALIFORNIA, USA / 28/11/2008 / 17/7/2009
43 / 235,338 / IN/PCT/2002/156/C HE / 10/07/2000 / 09/07/1999 / "A METHOD FOR MAKING A RECOMBINANT DNA" / THE EUROPEAN MOLECULAR BIOLOGY LABORATORY, GERMANY / 12/10/2007 / 17/7/2009
44 / 235,665 / 477/KOL/2005 / 07/06/2005 / 07/06/2004 / METHOD FOR MEDICAL 3D IMAGE DISPLAY AND PROCESSING, COMPUTER TO MOGRAPH AND WORKSTATION / SIEMENS AKTIENGESELLSCHAFT, GERMANY / 12/01/2007 / 31/7/2009
45 / 235,672 / 1942/KOLNP/2005 / 08/03/2004 / 06/03/2003 / AMYLASES, NUCLEIC ACIDS ENCODING THEM AND METHODS FOR MAKING AND USING THEM / VERENIUM CORPORATION, DIVERSA CORPORATION, USA / 30/03/2007 / 31/7/2009
46 / 235,674 / 1604/KOLNP/2004 / 22/04/2003 / 26/04/2002 / TACHYKININ RECEPTOR ANTAGONISTS / ELI LILLY AND COMPANY, USA / 11/08/2006 / 31/7/2009

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